[CAS NO. 119391-73-0] mAChR-IN-1hydrochloride

Name: mAChR-IN-1hydrochloride
Brand: Arctom Scientific
SKU: AS937433

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PRODUCTS SPECIFICATIONS [119391-73-0]

Distributor

Catalog

AS937433

Brand

Arctom Scientific

CAS

119391-73-0

MDL	-
Molecular Weight	524.82
Molecular Formula	C23H26ClIN2O2
SMILES	O=C(C(C1CCN(CC2=CC=C(I)C=C2)CC1)(C3=CC=CC=C3)CC4)NC4=O.[H]Cl

For research use only. We do not sell to patients.

mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC ₅₀ of 17 nM ^[1] .

IC50: 17 nM (mAChR) ^[1] .

Solid

Room temperature in continental US; may vary elsewhere.

4°C, sealed storage, away from moisture and light

* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

In Vitro:

DMSO : 65 mg/mL ( 123.85 mM ; Need ultrasonic)

H ₂ O : 1 mg/mL ( 1.91 mM ; ultrasonic and warming and heat to 60°C)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

* Please refer to the solubility information to select the appropriate solvent.

In Vivo:

1.

Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

Solubility: ≥ 2.17 mg/mL (4.13 mM); Clear solution
2.

Add each solvent one by one: 10% DMSO >> 90% (20% SBE-β-CD in saline)

Solubility: ≥ 2.17 mg/mL (4.13 mM); Clear solution
3.

Add each solvent one by one: 10% DMSO >> 90% corn oil

Solubility: ≥ 2.17 mg/mL (4.13 mM); Clear solution

* All of the co-solvents are available by MCE.