[CAS NO. 2110449-60-8] GlutaminylCyclaseInhibitor1

Name: GlutaminylCyclaseInhibitor1
Brand: Arctom Scientific
SKU: AS898037

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PRODUCTS SPECIFICATIONS [2110449-60-8]

Distributor

Catalog

AS898037

Brand

Arctom Scientific

CAS

2110449-60-8

MDL	MFCD31657434
Molecular Weight	369.43
Molecular Formula	C21H24FN3O2
SMILES	FC1=CC=CC(C2=CC(OC)=C(OC)C=C2)=C1NCCCN3C=C(C)N=C3

For research use only. We do not sell to patients.

Glutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor with an IC ₅₀ of 0.5 μM.

IC50: 0.5 μM (Glutaminyl cyclase) ^[1]

Glutaminyl Cyclase Inhibitor 1 is compound 23 ^[1] .

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Solid

Room temperature in continental US; may vary elsewhere.

In Vitro:

Ethanol : 100 mg/mL ( 270.69 mM ; Need ultrasonic)

DMSO : 83.33 mg/mL ( 225.56 mM ; Need ultrasonic)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

* Please refer to the solubility information to select the appropriate solvent.

In Vivo:

1.

Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

Solubility: ≥ 2.08 mg/mL (5.63 mM); Clear solution
2.

Add each solvent one by one: 10% DMSO >> 90% (20% SBE-β-CD in saline)

Solubility: ≥ 2.08 mg/mL (5.63 mM); Clear solution
3.

Add each solvent one by one: 10% DMSO >> 90% corn oil

Solubility: ≥ 2.08 mg/mL (5.63 mM); Clear solution

* All of the co-solvents are available by MCE.