[CAS NO. 2230850-47-0] EHMT2-IN-2
PRODUCTS SPECIFICATIONS [2230850-47-0]
DESCRIPTION [2230850-47-0]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 374.44 |
| Molecular Formula | C21H22N6O |
| SMILES | CC1=CC(NC)=NC(NC2=CC=C(OC)C(C(N3)=C(C)C4=C3C=NC=C4)=C2)=N1 |
Summary
IC50 & Target
|
EHMTI PEP <100 nM (IC 50 ) |
EHMT2 PEP <100 nM (IC 50 ) |
EHMT2 ICW <100 nM (IC 50 ) |
In Vitro
EHMT2-IN-2 (Compound 200) is a potent EHMT inhibitor, with IC 50 s of all < 100 nM for EEHMT1 peptide, EHMT2 peptide and cellular EHMT2 [1] .
MCE has not independently confirmed the accuracy of these methods. They are for reference only.
Appearance
Solid
Shipping
Room temperature in continental US; may vary elsewhere.
Storage
| Powder | -20°C | 3 years |
|---|---|---|
| 4°C | 2 years | |
| In solvent | -80°C | 6 months |
| -20°C | 1 month |
Solvent & Solubility
DMSO : 50 mg/mL ( 133.53 mM ; Need ultrasonic)
Stock Solutions
| Concentration Solvent Mass | 1 mg | 5 mg | 10 mg |
|---|
| 1 mM | 2.6707 mL | 13.3533 mL | 26.7065 mL |
| 5 mM | 0.5341 mL | 2.6707 mL | 5.3413 mL |
| 10 mM | 0.2671 mL | 1.3353 mL | 2.6707 mL |
