[CAS NO. 2235358-74-2]  Deltasonamide2(TFA)

Ships within Stock Price Qty Total
$0.00
$0.00
Please click "REQUEST A QUOTE" button if you need other sizes or custom synthesis
request a quote
If there is no stock, or you need other sizes or custom synthesis, please:

PRODUCTS SPECIFICATIONS [2235358-74-2]

Store
Catalog
AS945191
Brand
Arctom Scientific
CAS
2235358-74-2

DESCRIPTION [2235358-74-2]

Overview

MDL-
Molecular Weight761.27
Molecular FormulaC32H40ClF3N6O6S2
SMILESO=S(C1=CC=C(S(=O)(N(CC2=CC=C(Cl)C=C2)C3CCCC3)=O)C=C1)(N([C@H]4CC[C@H](N)CC4)CC5=NC(NC)=NC=C5)=O.O=C(O)C(F)(F)F

For research use only. We do not sell to patients.

1 Publications Citing Use of MCE


Summary

Deltasonamide 2 TFA is competitive, high affinity PDEδ inhibitor with a K d of ~385 pM [1] .


IC50 & Target

Kd: ~385 pM (PDEδ) [1]


Appearance

Solid


Shipping

Room temperature in continental US; may vary elsewhere.


Storage

4°C, sealed storage, away from moisture

* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)


Solvent & Solubility

In Vitro:

DMSO : 125 mg/mL ( 164.20 mM ; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.3136 mL 6.5680 mL 13.1359 mL
5 mM 0.2627 mL 1.3136 mL 2.6272 mL
10 mM 0.1314 mL 0.6568 mL 1.3136 mL
* Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

    Solubility: ≥ 2.08 mg/mL (2.73 mM); Clear solution

  • 2.

    Add each solvent one by one: 10% DMSO >> 90% corn oil

    Solubility: ≥ 2.08 mg/mL (2.73 mM); Clear solution

* All of the co-solvents are available by MCE.