[CAS NO. 330203-01-5] TC HSD 21
PRODUCTS SPECIFICATIONS [330203-01-5]
DESCRIPTION [330203-01-5]
Overview
| MDL | MFCD22683848 |
|---|---|
| Molecular Weight | 422.32 |
| Molecular Formula | C17H12BrNO3S2 |
| SMILES | O=C1N(C2=CC=C(OC)C=C2)C(S/C1=C\C3=CC=C(O)C(Br)=C3)=S |
Summary
TC HSD 21 is a potent 17β-hydroxysteroid dehydrogenase type 3 (17β-HSD3) inhibitor with an IC 50 of 14 nM. TC HSD 21 shows excellent selectivity over 17β-HSD isoenzymes and nuclear receptors [1] .
IC50 & Target
IC50: 14 nM (17β-HSD3) [1]
Appearance
Solid
Shipping
Room temperature in continental US; may vary elsewhere.
Storage
| Powder | -20°C | 3 years |
|---|---|---|
| 4°C | 2 years | |
| In solvent | -80°C | 6 months |
| -20°C | 1 month |
Solvent & Solubility
DMSO : ≥ 250 mg/mL ( 591.97 mM )
* "≥" means soluble, but saturation unknown.
Stock Solutions
| Concentration Solvent Mass | 1 mg | 5 mg | 10 mg |
|---|
| 1 mM | 2.3679 mL | 11.8394 mL | 23.6787 mL |
| 5 mM | 0.4736 mL | 2.3679 mL | 4.7357 mL |
| 10 mM | 0.2368 mL | 1.1839 mL | 2.3679 mL |
