[CAS NO. 372523-75-6] TCS-OX2-29

Name: TCS-OX2-29
Brand: Arctom Scientific
SKU: AS066547

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PRODUCTS SPECIFICATIONS [372523-75-6]

Distributor

Catalog

AS066547

Brand

Arctom Scientific

CAS

372523-75-6

DESCRIPTION [372523-75-6]

Overview

MDL	-
Molecular Weight	397.51
Molecular Formula	C23H31N3O3
SMILES	C([C@@H](NCC=1C=CN=CC1)C(C)(C)C)(=O)N2CC=3C(=CC(OC)=C(OC)C3)CC2

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

Concentration Volume Mass	1 mg	5 mg	10 mg
1 mM	2.5157 mL	12.5783 mL	25.1566 mL
5 mM	0.5031 mL	2.5157 mL	5.0313 mL
10 mM	0.2516 mL	1.2578 mL	2.5157 mL
50 mM	0.0503 mL	0.2516 mL	0.5031 mL

Description

TCX-OX2-29 is a antagonist (pKi = 7.5) that exhibits >250-fold selectivity for hOX2R compared with hOX1R (IC50s = 40 nM and >10,000 nM, respectively).

Synonyms

1-Butanone, 1-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-3,3-dimethyl-2-[(4-pyridinylmethyl)amino]-, (2S)-

Isoquinoline, 2-[(2S)-3,3-dimethyl-1-oxo-2-[(4-pyridinylmethyl)amino]butyl]-1,2,3,4-tetrahydro-6,7-dimethoxy-

(2S)-1-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-3,3-dimethyl-2-[(4-pyridinylmethyl)amino]-1-butanone

(2S)-2-(4-Pyridylmethylamino)-1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3,3-dimethylbutan-1-one

TCS-OX 2-29

TCS-OX2-29

Orexin antagonist TCS-OX2-29