[CAS NO. 794568-90-4]  BAY 73-6691 racemate

Ships within Stock Price Qty Total
$0.00
$0.00
Please click "REQUEST A QUOTE" button if you need other sizes or custom synthesis
request a quote
If there is no stock, or you need other sizes or custom synthesis, please:

PRODUCTS SPECIFICATIONS [794568-90-4]

Store
Catalog
AS904602
Brand
Arctom Scientific
CAS
794568-90-4

DESCRIPTION [794568-90-4]

Overview

MDLMFCD31619335
Molecular Weight356.73
Molecular FormulaC15H12ClF3N4O
SMILESO=C1C2=C(N(C3=CC=CC=C3Cl)N=C2)NC(CC(C)C(F)(F)F)=N1

For research use only. We do not sell to patients.

Summary

BAY 73-6691 racemate is a phosphodiesterase 9 inhibitor extracted from patent WO 2017070293 A1.


IC50 & Target

phosphodiesterase 9 [1]


Appearance

Solid


Shipping

Room temperature in continental US; may vary elsewhere.


Storage

Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month

Solvent & Solubility

In Vitro:

DMSO : ≥ 100 mg/mL ( 280.32 mM )

* "≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.8032 mL 14.0162 mL 28.0324 mL
5 mM 0.5606 mL 2.8032 mL 5.6065 mL
10 mM 0.2803 mL 1.4016 mL 2.8032 mL
* Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

    Solubility: 5 mg/mL (14.02 mM); Clear solution; Need ultrasonic

  • 2.

    Add each solvent one by one: 10% DMSO >> 90% (20% SBE-β-CD in saline)

    Solubility: 5 mg/mL (14.02 mM); Suspended solution; Need ultrasonic

  • 3.

    Add each solvent one by one: 10% DMSO >> 90% corn oil

    Solubility: 5 mg/mL (14.02 mM); Clear solution; Need ultrasonic

* All of the co-solvents are available by MCE.