[CAS NO. 86434-57-3]  Beperidium iodide

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PRODUCTS SPECIFICATIONS [86434-57-3]

Distributor
Catalog
AS257663
Brand
Arctom Scientific
CAS
86434-57-3

DESCRIPTION [86434-57-3]

Overview

MDLMFCD00866899
Molecular Weight527.44
Molecular FormulaC23H34IN3O3
SMILESC[N+]1(CC)CCC(OC(C(C2=NOC3=C2C=CC=C3)N4CCCCCC4)=O)CC1.[I-]

For research use only. We do not sell to patients.

Summary

Beperidium iodide shows a competitive antagonistic effect against acetylcholine receptor with a pA2 of 7.93.


IC50 & Target

pA2: 7.93 (Acetylcholine receptor) [1]


Appearance

Solid


Shipping

Room temperature in continental US; may vary elsewhere.


Storage

4°C, sealed storage, away from moisture and light

* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)


Solvent & Solubility

In Vitro:

DMSO : ≥ 100 mg/mL ( 189.60 mM )

* "≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.8960 mL 9.4798 mL 18.9595 mL
5 mM 0.3792 mL 1.8960 mL 3.7919 mL
10 mM 0.1896 mL 0.9480 mL 1.8960 mL
* Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

    Solubility: ≥ 2.5 mg/mL (4.74 mM); Clear solution

  • 2.

    Add each solvent one by one: 10% DMSO >> 90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (4.74 mM); Clear solution

  • 3.

    Add each solvent one by one: 10% DMSO >> 90% corn oil

    Solubility: ≥ 2.5 mg/mL (4.74 mM); Clear solution

* All of the co-solvents are available by MCE.