[CAS NO. 2098884-52-5] Lenumlostat

Name: Lenumlostat
Brand: Arctom Scientific
SKU: AS1021851

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PRODUCTS SPECIFICATIONS [2098884-52-5]

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Catalog

AS1021851

Brand

Arctom Scientific

CAS

2098884-52-5

DESCRIPTION [2098884-52-5]

Overview

MDL	-
Molecular Weight	399.34
Molecular Formula	C18H17F4N3O3
SMILES	FC(F)(C1=NC(OC2=CC(C(N(C[C@H]3O)C[C@H]3F)=O)=CC=C2)=CC(CN)=C1)F

For research use only. We do not sell to patients.

Summary

Lenumlostat is a Lysyl Oxidase Like 2 (LOXL2) inhibitor with an IC ₅₀ value <300 nM. Lenumlostat also exhibits antifibrotic activity ^[1] ^[2] .

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Room temperature in continental US; may vary elsewhere.

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Please store the product under the recommended conditions in the Certificate of Analysis.

References

[1] Lonergan David, et al. Preparation of aminomethyltrifluoromethylpyridinyloxyphenylfluorohydroxypyrrolidinylmethanone derivatives for use as lysyl oxidase-like 2 inhibitors: World Intellectual Property Organization, WO2018048943. 2018-03-15.
[2] WHO Drug Information-World Health Organization (WHO).