[CAS NO. 23672-07-3] Levosulpiride

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PRODUCTS SPECIFICATIONS [23672-07-3]

Catalog

AS437336

Brand

Arctom Scientific

CAS

23672-07-3

DESCRIPTION [23672-07-3]

Overview

MDL	MFCD00055220
Molecular Weight	341.43
Molecular Formula	C15H23N3O4S
SMILES	O=C(NC[C@H]1N(CC)CCC1)C2=CC(S(=O)(N)=O)=CC=C2OC

For research use only. We do not sell to patients.

Summary

Levosulpiride (RV-12309) is the (S)-enantiomer of sulpiride, which is a D2 receptor a antagonist, an atypical antipsychotic drug of the benzamide class.

Clinical Trial

NCT Number	Sponsor	Condition	Start Date	Phase
NCT02481583	Wuhan Union Hospital, China	Dyspepsia	March 2013	Phase 1
NCT03161652	Carmen Clapp\|Instituto Mexicano de Oftalmologia (IMO)\|Universidad Autónoma de Querétaro\|General Hospital Nuremberg & Paracelsus Medical University Nuremberg\|Instituto de la Retina del Bajio SC (INDEREB)\|Instituto de Neurobiología, Universidad Nacional Autonoma de Mexico (UNAM)\|Universidad Nacional Autonoma de Mexico	Diabetic Macular Edema\|Diabetic Retinopathy	May 24, 2017	Phase 2
NCT00866645	Shanghai Mental Health Center\|Shanghai Hotmed Sciences Co.,LTD	Agitation	February 2009	Phase 2\|Phase 3
NCT04697641	Sir Ganga Ram Hospital	Dyspepsia\|Helicobacter Pylori Infection	September 1, 2017	Not Applicable

Appearance

Solid

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

Solvent & Solubility

In Vitro:

DMSO : 50 mg/mL ( 146.44 mM ; Need ultrasonic)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.9289 mL	14.6443 mL	29.2886 mL
5 mM	0.5858 mL	2.9289 mL	5.8577 mL
10 mM	0.2929 mL	1.4644 mL	2.9289 mL

* Please refer to the solubility information to select the appropriate solvent.

In Vivo:

1.

Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

Solubility: ≥ 2.5 mg/mL (7.32 mM); Clear solution
2.

Add each solvent one by one: 10% DMSO >> 90% (20% SBE-β-CD in saline)

Solubility: ≥ 2.5 mg/mL (7.32 mM); Clear solution
3.

Add each solvent one by one: 10% DMSO >> 90% corn oil

Solubility: ≥ 2.5 mg/mL (7.32 mM); Clear solution

* All of the co-solvents are available by MCE.

Synonyms

Benzamide, 5-(aminosulfonyl)-N-[[(2S)-1-ethyl-2-pyrrolidinyl]methyl]-2-methoxy-

o-Anisamide, N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-sulfamoyl-, (-)-

Benzamide, 5-(aminosulfonyl)-N-[(1-ethyl-2-pyrrolidinyl)methyl]-2-methoxy-, (S)-

5-(Aminosulfonyl)-N-[[(2S)-1-ethyl-2-pyrrolidinyl]methyl]-2-methoxybenzamide

l-Sulpiride

(-)-Sulpiride

L-Sulpiride

S-(-)-Sulpiride

S-Sulpiride

Levosulpiride

Levobren

Levopraid

sulpid

levopride

Lesuride