Overview
| MDL | - |
|---|
| Molecular Weight | 353.4 |
|---|
| Molecular Formula | C18H15N3O3S |
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| SMILES | - |
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For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg |
| 1 mM | 2.8297 mL | 14.1483 mL | 28.2965 mL |
| 5 mM | 0.5659 mL | 2.8297 mL | 5.6593 mL |
| 10 mM | 0.2830 mL | 1.4148 mL | 2.8297 mL |
| 50 mM | 0.0566 mL | 0.2830 mL | 0.5659 mL |
Description
NI-42 is a biased, potent inhibitor of the of the with IC50s of 7.9, 48, 260 nM for BRPF1/2/3.
Targets
BRPF1 [1] (in the BROMOscan assay) | BRPF2 [1] (in the BROMOscan assay) | BRPF3 [1] (in the BROMOscan assay) |
| 7.9 nM | 48 nM | 260 nM |