| MDL | - |
|---|---|
| Molecular Weight | 430.59 |
| Molecular Formula | C21H26N4O2S2 |
| SMILES | O=S(C1=CC=C(C2=CSC=C2)C=C1)(N3C(N4CCN(C5CCC5)CC4)=NCC3)=O |
KDM2B-IN-2, a potent histone demethylase (kdm2b) inhibitor with an IC 50 of 0.021 μM in a KDM2B TR-FRET assay. KDM2B-IN-2 can be used for hyperproliferative diseases research [1] .
|
KDM2B 0.021 μM (IC 50 ) |
Solid
Room temperature in continental US; may vary elsewhere.
| Powder | -20°C | 3 years |
|---|---|---|
| 4°C | 2 years | |
| In solvent | -80°C | 6 months |
| -20°C | 1 month |
DMSO : 31.25 mg/mL ( 72.57 mM ; ultrasonic and heat to 80°C)
| Concentration Solvent Mass | 1 mg | 5 mg | 10 mg |
|---|
| 1 mM | 2.3224 mL | 11.6120 mL | 23.2239 mL |
| 5 mM | 0.4645 mL | 2.3224 mL | 4.6448 mL |
| 10 mM | 0.2322 mL | 1.1612 mL | 2.3224 mL |