[CAS NO. ] Nociceptin (1-13), amide TFA

Name: Nociceptin (1-13), amide TFA
Brand: Arctom Scientific
SKU: HY-P1317A

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PRODUCTS SPECIFICATIONS

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Catalog

HY-P1317A

Brand

MCE

CAS

-

DESCRIPTION

Overview

MDL	-
Molecular Weight	1495.61
Molecular Formula	C63H101F3N22O17
SMILES	-

For research use only. We do not sell to patients.

Summary

Nociceptin (1-13), amide TFA is a potent ORL1 receptor (opioid receptor-like 1 receptor, OP4) agonist with a pEC ₅₀ of 7.9 for mouse vas deferens and a K _i of 0.75 nM for binding to rat forebrain membranes ^[1] ^[2] .

Appearance

Solid

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Sealed storage, away from moisture

Powder	-80°C	2 years
	-20°C	1 year

* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility

In Vitro:

DMSO : ≥ 100 mg/mL ( 66.86 mM )

* "≥" means soluble, but saturation unknown.

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	0.6686 mL	3.3431 mL	6.6862 mL
5 mM	0.1337 mL	0.6686 mL	1.3372 mL
10 mM	0.0669 mL	0.3343 mL	0.6686 mL

* Please refer to the solubility information to select the appropriate solvent.

In Vivo:

1.

Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

Solubility: ≥ 2.5 mg/mL (1.67 mM); Clear solution
2.

Add each solvent one by one: 10% DMSO >> 90% (20% SBE-β-CD in saline)

Solubility: ≥ 2.5 mg/mL (1.67 mM); Clear solution
3.

Add each solvent one by one: 10% DMSO >> 90% corn oil

Solubility: ≥ 2.5 mg/mL (1.67 mM); Clear solution

* All of the co-solvents are available by MCE.