[CAS NO. 150322-43-3] Prasugrel

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PRODUCTS SPECIFICATIONS [150322-43-3]

Catalog

SLK-S1258

Brand

Selleck

CAS

150322-43-3

DESCRIPTION [150322-43-3]

Overview

MDL	MFCD09954140
Molecular Weight	373.44
Molecular Formula	C20H20FNO3S
SMILES	C(C(=O)C1CC1)(N2CC3=C(CC2)SC(OC(C)=O)=C3)C4=C(F)C=CC=C4

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

Concentration Volume Mass	1 mg	5 mg	10 mg
1 mM	2.6778 mL	13.3890 mL	26.7781 mL
5 mM	0.5356 mL	2.6778 mL	5.3556 mL
10 mM	0.2678 mL	1.3389 mL	2.6778 mL
50 mM	0.0536 mL	0.2678 mL	0.5356 mL

Description

Prasugrel (Effient, Efient, Prasita,CS-747, LY640315,PCR 4099) is a thienopyridine antagonist, used for the reduction of thrombotic cardiovascular events.

Targets

P2Y12 receptor ^[1]

In vitro

Prasugrel is a novel orally active thienopyridine with faster, higher and more reliable inhibition of platelet aggregation than clopidogrel reflecting its metabolism in vivo to an active metabolite with selective P2Y(12) antagonistic activity.

References

[1] Hashimoto M, et al. Biochem Pharmacol, 2007, 74(7), 1003-1009.
[2] Ogawa T, et al. Eur J Pharmacol, 2009, 612(1-3), 29-34.
[3] Niitsu Y, et al. Eur J Pharmacol, 2008, 579(1-3), 276-282.

Synonyms

Ethanone, 2-[2-(acetyloxy)-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl]-1-cyclopropyl-2-(2-fluorophenyl)-

Thieno[3,2-c]pyridine, ethanone deriv.

2-[2-(Acetyloxy)-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl]-1-cyclopropyl-2-(2-fluorophenyl)ethanone

CS 747

Prasugrel

2-Acetoxy-5-(α-cyclopropylcarbonyl-2-fluorobenzyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridine

LY 640315

Effient free base

2-Acetoxy-5-(α-cyclopropylcarbonyl-2-fluorobenzyl)-4,5,6,7-tetrahydrothieno-[3,2-c]pyridine

[5-[2-Cyclopropyl-1-(2-fluorophenyl)-2-oxoethyl]-6,7-dihydro-4H-thieno[3,2-c]pyridin-2-yl] acetate