[CAS NO. 97792-45-5] Lappaconite HBr

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PRODUCTS SPECIFICATIONS [97792-45-5]

Catalog

SLK-S2387

Brand

Selleck

CAS

97792-45-5

DESCRIPTION [97792-45-5]

Overview

MDL	-
Molecular Weight	665.61
Molecular Formula	C32H44N2O8.HBr
SMILES	O(C)[C@@H]1[C@]23[C@H]4[C@](OC(=O)C5=C(NC(C)=O)C=CC=C5)(CN(CC)[C@@]2([C@H](C4)[C@]6(O)[C@]7(O)[C@]3(C[C@@H]([C@@H]7OC)[C@@H](OC)C6)[H])[H])CC1.Br

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

Concentration Volume Mass	1 mg	5 mg	10 mg
1 mM	1.5024 mL	7.5119 mL	15.0238 mL
5 mM	0.3005 mL	1.5024 mL	3.0048 mL
10 mM	0.1502 mL	0.7512 mL	1.5024 mL
50 mM	0.0300 mL	0.1502 mL	0.3005 mL

Description

Lappaconite Hydrobromide is a kind of alkaloid extracted from Aconitum sinomontanum Nakai and has anti-inflammatory effects.

In vitro

Lappaconite Hydrobromide is a kind of alkaloid extracted from Aconitum sinomontanum Nakai and has anti-inflammatory effects. Its absorption percentage in rat stomachs after administration was 9.67%.The absorption percentages at duodenum,jejunum,ileum and colon were 19.61%,11.83%,12.95% and 9.51%, respectively.When the concentration was raised from 10 mg/L to 40 mg/L, the uptake of lappaconite hydrobromide was linearly increased,whereas the absorption rate constant kept at the same level.

In vivo

LD50: Mice 10.5mg/kg (i.p.); Rats 9.9mg/kg (i.p.)

Synonyms

Aconitane-4,8,9-triol, 20-ethyl-1,14,16-trimethoxy-, 4-[2-(acetylamino)benzoate], hydrobromide (1:1), (1α,14α,16β)-

Aconitane-4,8,9-triol, 20-ethyl-1,14,16-trimethoxy-, 4-[2-(acetylamino)benzoate], monohydrobromide, (1α,14α,16β)-

2H-12,3,6a-Ethanylylidene-7,9-methanonaphth[2,3-b]azocine, aconitane-4,8,9-triol deriv.

Lappaconitine hydrobromide

Allapinine

Allafort