Overview
| MDL | - |
|---|
| Molecular Weight | 417.54 |
|---|
| Molecular Formula | C27H31NO3 |
|---|
| SMILES | - |
|---|
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg |
| 1 mM | 2.3950 mL | 11.9749 mL | 23.9498 mL |
| 5 mM | 0.4790 mL | 2.3950 mL | 4.7900 mL |
| 10 mM | 0.2395 mL | 1.1975 mL | 2.3950 mL |
| 50 mM | 0.0479 mL | 0.2395 mL | 0.4790 mL |
Description
GSK5182, 4-hydroxytamoxifen analog, is a specific inverse agonist of that inhibits pro-inflammatory cytokine-induced catabolic factors.
In vitro
GSK5182, a small-molecule ERRγ inverse agonist, inhibits pro-inflammatory cytokine-induced catabolic factors in mouse articular chondrocytes.