[CAS NO. 1135242-13-5]  VU0357017 Hydrochloride

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PRODUCTS SPECIFICATIONS [1135242-13-5]

Distributor
Catalog
SLK-S6795
Brand
Selleck
CAS
1135242-13-5

DESCRIPTION [1135242-13-5]

Overview

MDLMFCD17215959
Molecular Weight369.89
Molecular FormulaC18H28ClN3O3
SMILESO=C(N1CCC(NCCNC(C2=CC=CC=C2C)=O)CC1)OCC.[H]Cl

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

1 mg5 mg10 mg
1 mM2.7035 mL13.5175 mL27.0351 mL
5 mM0.5407 mL2.7035 mL5.4070 mL
10 mM0.2704 mL1.3518 mL2.7035 mL
50 mM0.0541 mL0.2704 mL0.5407 mL

Description

VU0357017 hydrochloride (CID-25010775) is a potent, highly selective and CNS-penetrant agonist of which is a subtype of . VU0357017 hydrochloride appears to act at an allosteric site to activate the receptor with EC50 of 477 nM and Ki of 9.91 μM.

Targets

M1 mAChR [1]
(Cell-free assay)
M1 mAChR [1]
(Cell-free assay)
477 nM(EC50)9.91 μM(Ki)