[CAS NO. 2071195-74-7]  Epertinib hydrochloride

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PRODUCTS SPECIFICATIONS [2071195-74-7]

Catalog
SLK-S6897
Brand
Selleck
CAS
2071195-74-7

DESCRIPTION [2071195-74-7]

Overview

MDL-
Molecular Weight596.48
Molecular FormulaC30H28Cl2FN5O3
SMILES-

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

1 mg5 mg10 mg
1 mM1.6765 mL8.3825 mL16.7650 mL
5 mM0.3353 mL1.6765 mL3.3530 mL
10 mM0.1677 mL0.8383 mL1.6765 mL
50 mM0.0335 mL0.1677 mL0.3353 mL

Description

Epertinib hydrochloride (S-222611 hydrochloride) is a potent, orally active, reversible, and selective inhibitor of , and with IC50 of 1.48 nM, 7.15 nM and 2.49 nM, respectively. Epertinib hydrochloride (S-222611 hydrochloride) exhibits antitumor activity.

Targets

EGFR [1]
(Cell-free assay)
HER4 [1]
(Cell-free assay)
HER2 [1]
(Cell-free assay)
1.48 nM2.49 nM7.15 nM