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[CAS NO. 1373625-34-3] ARN077
| Ships within | Stock | Price | Qty | Total |
Please click "REQUEST A QUOTE" button if there is no stock, or you need other sizes or custom synthesis.
| Catalog: | HY-120813 |
| Brand: | MCE |
| CAS: | 1373625-34-3 |
Overview
| MDL | - |
|---|---|
| Molecular Weight | 291.34 |
| Molecular Formula | C16H21NO4 |
| SMILES | O=C(OCCCCCC1=CC=CC=C1)N[C@@H]2[C@H](C)OC2=O |
Summary
IC50 & Target
IC50: 7 nM (human NAAA) [1] .
Appearance
Solid
Shipping
Room temperature in continental US; may vary elsewhere.
Storage
| Powder | -20°C | 3 years |
|---|---|---|
| 4°C | 2 years | |
| In solvent | -80°C | 6 months |
| -20°C | 1 month |
Solvent & Solubility
DMSO : 250 mg/mL ( 858.10 mM ; Need ultrasonic)
Stock Solutions
| Concentration Solvent Mass | 1 mg | 5 mg | 10 mg |
|---|
| 1 mM | 3.4324 mL | 17.1621 mL | 34.3242 mL |
| 5 mM | 0.6865 mL | 3.4324 mL | 6.8648 mL |
| 10 mM | 0.3432 mL | 1.7162 mL | 3.4324 mL |
References
- [1] Sasso O, et al. Antinociceptive effects of the N-acylethanolamine acid amidase inhibitor ARN077 in rodent pain models. Pain. 2013 Mar;154(3):350-60.
- [2] Davis MP, et al. Cannabinoids in pain management: CB1, CB2 and non-classic receptor ligands. Expert Opin Investig Drugs. 2014 Aug;23(8):1123-40.
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