[CAS NO. 2244451-48-5] BI-4916
PRODUCTS SPECIFICATIONS [2244451-48-5]
DESCRIPTION [2244451-48-5]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 527.42 |
| Molecular Formula | C23H24Cl2N2O6S |
| SMILES | O=C(OCC)CS(=O)(C1=CC=C([C@H](NC(C(N2C)=CC3=C2C=C(C)C(Cl)=C3Cl)=O)CO)C=C1)=O |
2 Publications Citing Use of MCE
Summary
BI-4916 is a prodrug of BI-4924. BI-4924 is a NADH/NAD + -competitive PHGDH inhibitor [1] .
Appearance
Solid
Shipping
Room temperature in continental US; may vary elsewhere.
Storage
| Powder | -20°C | 3 years |
|---|---|---|
| 4°C | 2 years | |
| In solvent | -80°C | 6 months |
| -20°C | 1 month |
Solvent & Solubility
DMSO : 250 mg/mL ( 474.01 mM ; Need ultrasonic)
Stock Solutions
| Concentration Solvent Mass | 1 mg | 5 mg | 10 mg |
|---|
| 1 mM | 1.8960 mL | 9.4801 mL | 18.9602 mL |
| 5 mM | 0.3792 mL | 1.8960 mL | 3.7920 mL |
| 10 mM | 0.1896 mL | 0.9480 mL | 1.8960 mL |
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1.
Add each solvent one by one: 10% DMSO >> 90% corn oil
Solubility: ≥ 2.08 mg/mL (3.94 mM); Clear solution