[CAS NO. 2376334-75-5] DS08210767
PRODUCTS SPECIFICATIONS [2376334-75-5]
DESCRIPTION [2376334-75-5]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 513.67 |
| Molecular Formula | C31H39N5O2 |
| SMILES | CC1(N=C(C2=CC=C(C=C2N(C1=O)C3=CC=C(C=C3)NCCNC4CCOCC4)C#N)C5CCCCC5)C |
Summary
DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC 50 of 90 nM [1] .
IC50 & Target
IC50: 90 nM (PTHR1) [1]
Appearance
Solid
Shipping
Room temperature in continental US; may vary elsewhere.
Storage
| Powder | -20°C | 3 years |
|---|---|---|
| In solvent | -80°C | 6 months |
| -20°C | 1 month |
Solvent & Solubility
DMSO : 5 mg/mL ( 9.73 mM ; ultrasonic and warming and heat to 80°C)
Stock Solutions
| Concentration Solvent Mass | 1 mg | 5 mg | 10 mg |
|---|
| 1 mM | 1.9468 mL | 9.7339 mL | 19.4678 mL |
| 5 mM | 0.3894 mL | 1.9468 mL | 3.8936 mL |
| 10 mM | --- | --- | --- |