[CAS NO. 2512847-06-0] LANA-DNA-IN-1
PRODUCTS SPECIFICATIONS [2512847-06-0]
DESCRIPTION [2512847-06-0]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 330.34 |
| Molecular Formula | C19H14N4O2 |
| SMILES | CC1=CC2=C(C=NC=C2C=C1)N3C=C(N=N3)C4=CC=C(C=C4)C(O)=O |
Summary
IC50 & Target
IC50: 8 μM (LBS2); 9μM LBS1); 8 μM (LBS3); 53 μM (wild-type LANA) [1]
In Vitro
LANA-DNA-IN-1 has inhibition activity for LBS2, LBS1 and LBS3 with IC
50
values of 8 μM, 9μM and 8μM in FP Assay
[1]
.
LANA-DNA-IN-1 has potent LANA-LBS1-inhibitory with an IC
50
values of 53 μM
[1]
.
LANA-DNA-IN-1 (31.25, 62.5, 125 and 250 μM) has potent against wild-type LANA CTD and the oligomerization-deficient LANA DBD mutant
[1]
.
MCE has not independently confirmed the accuracy of these methods. They are for reference only.
Shipping
Room temperature in continental US; may vary elsewhere.
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.