[CAS NO. 341944-06-7] Antibacterial agent 117
PRODUCTS SPECIFICATIONS [341944-06-7]
DESCRIPTION [341944-06-7]
Overview
| MDL | MFCD00215049 |
|---|---|
| Molecular Weight | 240.71 |
| Molecular Formula | C9H9ClN4S |
| SMILES | NC1=NNC(SCC2=CC=CC=C2Cl)=N1 |
Summary
IC50 & Target
IC50: 15 μM (RpMetAP1) [1]
In Vitro
Antibacterial agent 117 can inhibit RpMetAP1 with an
IC
50
value of 15 μM
[1]
.
Antibacterial agent 117 (0.3 μM, 3 μM, 30 μM and 300 μM) stimulates endothelial cell (EC) metabolism and also inhibits rickettsial growth
[1]
.
MCE has not independently confirmed the accuracy of these methods. They are for reference only.
Appearance
Solid
Shipping
Room temperature in continental US; may vary elsewhere.
Storage
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
Solvent & Solubility
DMSO : 100 mg/mL ( 415.44 mM ; Need ultrasonic)
Stock Solutions
| Concentration Solvent Mass | 1 mg | 5 mg | 10 mg |
|---|
| 1 mM | 4.1544 mL | 20.7719 mL | 41.5438 mL |
| 5 mM | 0.8309 mL | 4.1544 mL | 8.3088 mL |
| 10 mM | 0.4154 mL | 2.0772 mL | 4.1544 mL |