Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
1 mg
5 mg
10 mg
1 mM
2.6497 mL
13.2485 mL
26.4971 mL
5 mM
0.5299 mL
2.6497 mL
5.2994 mL
10 mM
0.2650 mL
1.3249 mL
2.6497 mL
50 mM
0.0530 mL
0.2650 mL
0.5299 mL
Description
GSK2982772 is an ATP competitive inhibitor with the IC50 value of 16 nM. It has exquisite kinase specificity and excellent activity in blocking many TNF-dependent cellular responses.
GSK2982772 has excellent activity in both RIP1 cellular systems, preventing TNF induced necrotic cell death, and an ulcerative colitis explant assay blocking spontaneous cytokine release.
